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Syntheses of optically pure β-hydroxyaspartate derivatives as glutamate transporter blockers

Keiko Shimamoto, Yasushi Shigeri, Yoshimi Yasuda‐Kamatani, Bruno Lebrun, Noboru Yumoto, Terumi Nakajima

Bioorganic & Medicinal Chemistry Letters · 2000 · 112 citations · 11 references

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11

Flux coupling in a neuronal glutamate transporter

Noa Zerangue, Michael P. Kavanaugh · Nature · 1996 · 858 citations

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dl-threo-β-Benzyloxyaspartate, A Potent Blocker of Excitatory Amino Acid Transporters

Keiko Shimamoto, Bruno Lebrun, Yoshimi Yasuda‐Kamatani et al. · Molecular Pharmacology · 1998 · 552 citations · Full text

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Conformationally defined neurotransmitter analogs. Selective inhibition of glutamate uptake by one pyrrolidine-2,4-dicarboxylate diastereomer

Richard J. Bridges, Mark Stanley, Michael W. Anderson et al. · Journal of Medicinal Chemistry · 1991 · 303 citations

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Contrasting Modes of Action of Methylglutamate Derivatives on the Excitatory Amino Acid Transporters, EAAT1 and EAAT2

Robert J. Vandenberg, Ann D. Mitrovic, Mary Chebib et al. · Molecular Pharmacology · 1997 · 106 citations

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New β-Hydroxyaspartate Derivatives Are Competitive Blockers for the Bovine Glutamate/Aspartate Transporter

Bruno Lebrun, Masahiro Sakaitani, Keiko Shimamoto et al. · Journal of Biological Chemistry · 1997 · 73 citations · Full text

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