Nature Biotechnology · 2015 · 350 citations · 44 references
PharmacyMedicinal ChemistryOncologyDrug DesignDrug DiscoveryMolecular OncologyChemical Probe DiscoveryProtein Kinase CascadesCancer Cell Proliferation InhibitionCell Proliferation SignalingEnzyme Target ValidationKinase Inhibitor Library DesignKinase InhibitorsKinase ProbesProtein Kinase InhibitorsTargeted Kinase Inhibition
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Specificity and mechanism of action of some commonly used protein kinase inhibitors
Stephen Davies, Helen Reddy, Matilde Caivano et al. · Biochemical Journal · 2000 · 4.1K citations · Full text
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Specificity and mechanism of action of some commonly used protein kinase inhibitors
Stephen Davies, Helen Reddy, Matilde Caivano et al. · Biochemical Journal · 2000 · 3.1K citations
The selectivity of protein kinase inhibitors: a further update
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A quantitative analysis of kinase inhibitor selectivity
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