Concepedia

Development of Potent and Selective Tissue Transglutaminase Inhibitors: Their Effect on TG2 Function and Application in Pathological Conditions

Eduard Badarau, Daniel L. Rathbone, Andrea Costanzi, Thomas Thibault, Colin E. Murdoch, Saı̈d El Alaoui, Milda Bartkeviciute, Martin Griffin

Chemistry & Biology · 2015 · 56 citations · 36 references

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36

Program DYNAFIT for the Analysis of Enzyme Kinetic Data: Application to HIV Proteinase

Petr Kuzmič · Analytical Biochemistry · 1996 · 1.5K citations

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Direct Evidence for the Presence of Histidine in the Active Center of Chymotrypsin<sup>*</sup>

Guenther Schoellmann, Elliott Shaw · Biochemistry · 1963 · 643 citations

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Transglutaminase 2 Undergoes a Large Conformational Change upon Activation

Daniel M. Pinkas, Pavel Strop, Axel T. Brünger et al. · PLoS Biology · 2007 · 445 citations · Full text

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Structural basis for the guanine nucleotide-binding activity of tissue transglutaminase and its regulation of transamidation activity

Shenping Liu, Richard A. Cerione, Jon Clardy · Proceedings of the National Academy of Sciences · 2002 · 314 citations · Full text

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DynaFit—A Software Package for Enzymology

Petr Kuzmič · Methods in enzymology on CD-ROM/Methods in enzymology · 2009 · 257 citations

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