Publication | Closed Access
A synthesis, in silico, in vitro and in vivo study of thieno[2,3-b]pyridine anticancer analogues
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Citations
36
References
2015
Year
Vivo StudyMedicinal ChemistryNatural SciencesMedicineMolecular BiologyPharmacological AgentOrganic ChemistryAnti-cancer AgentQuantum ChemistryChemistrySupramolecular ChemistryPharmacologyHeterocycle ChemistryMolecular ChemistrySynthetic ChemistryDrug Discovery
The thieno[2,3-<italic>b</italic>]pyridines bind to TDP1 with the best analogue <bold>9d</bold> with IC<sub>50</sub> at 0.5 μM.
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