Discovery of a Small‐Molecule Inhibitor of the KIX–KID Interaction

Abstract

Are you too small? The small molecule (MW=297) shown here was discovered to be an inhibitor of the KIX–KID interaction by using a novel Renilla luciferase complementation assay. This compound also inhibits CREB-mediated gene transcription in living cells. Detailed facts of importance to specialist readers are published as ”Supporting Information”. Such documents are peer-reviewed, but not copy-edited or typeset. They are made available as submitted by the authors. Please note: The publisher is not responsible for the content or functionality of any supporting information supplied by the authors. Any queries (other than missing content) should be directed to the corresponding author for the article.