Kinetic Selectivity Analysis

Kinetic Selectivity Analysis is a quantitative method in covalent drug design that distinguishes target engagement specificity by measuring the relative rates of covalent bond formation between a drug and competing off-target proteins under physiological conditions.

68

Publications

3.1K

Citations

331

Authors

118

Institutions

Publications per year

2017–2026

23

Authors

331

  1. DJ
    David J. Mann

    Imperial College London, United Kingdom

    3 publications · 111 citations

    3

    h-index

  2. RM
    Rhodri M. L. Morgan

    Imperial College London, United Kingdom

    3 publications · 111 citations

    3

    h-index

  3. WW
    William W. Brennessel

    University of Rochester, United States

    3 publications · 262 citations

    3

    h-index

  4. AA
    Alan Armstrong

    Imperial College London, United Kingdom

    3 publications · 111 citations

    3

    h-index

  5. DP
    Dominic P. Affron

    Imperial College London, United Kingdom

    3 publications · 111 citations

    3

    h-index

1–5 of 331

Venues

  1. Journal of the American Chemical Society

    JACS · 13 publications · 1.1K citations

    13

    h-index

  2. Organometallics

    5 publications · 231 citations

    5

    h-index

  3. Chemical Engineering Journal

    3 publications · 138 citations

    3

    h-index

  4. Organic & Biomolecular Chemistry

    3 publications · 64 citations

    3

    h-index

  5. Industrial & Engineering Chemistry Research

    3 publications · 132 citations

    3

    h-index

1–5