Dinesh Gala

Preparations of antifungal Sch 42427/SM 9164: Preparative chromatographic resolution, and total asymmetric synthesis via enzymatic preparation of chiral α-hydroxy arylketones

Dinesh Gala, Donald J. DiBenedetto, Jon E. Clark et al. · Tetrahedron Letters · 1996 · 63 citations

Antifungal Agent, Total Asymmetric Synthesis, Antifungal Agents +6

Antitumor Imidazotetrazines. 35. New Synthetic Routes to the Antitumor Drug Temozolomide

Yongfeng Wang, Malcolm F. G. Stevens, Tze‐Ming Chan et al. · The Journal of Organic Chemistry · 1997 · 34 citations

Organic Chemistry, Pharmacotherapy, Heterocycle Chemistry +17

Mono N-arylation of piperazine(III): metal-catalyzed N-arylation and its application to the novel preparations of the antifungal posaconazole and its advanced intermediate

Michael Hepperle, Jeffrey Eckert, Dinesh Gala et al. · Tetrahedron Letters · 2002 · 32 citations

Antifungal Posaconazole, Antifungal Agent, Mono N-arylation +4

Sequential mono-N-arylation of piperazine nitrogens. Part 1: A simplified method and its application to the preparation of a key N,N′-biaryl piperazine antifungal intermediate

Michael Hepperle, Jeffrey Eckert, Dinesh Gala · Tetrahedron Letters · 1999 · 27 citations

Antifungal Agent, Sequential Mono-n-arylation, Piperazine Nitrogens +4

A convenient, improved synthesis of (camphoryl)sulfonyl oxaziridines.

Ingrid Mergelsberg, Dinesh Gala, Dominik Scherer et al. · Tetrahedron Letters · 1992 · 27 citations

Organic Chemistry, Sulfonyl Oxaziridines, Synthetic Chemistry +1