Pyrrole-singlet oxygen reactions leading to α,α′-bipyrroles. Synthesis of prodigiosin and analogs

Harry H. Wasserman, Anders K. Petersen, Mingde Xia, +1

Tetrahedron Letters

EngineeringBiochemistrySinglet OxygenNatural SciencesOrganic Chemistry +8

Application of acyl cyanophosphorane methodology to the synthesis of protease inhibitors: poststatin, eurystatin, phebestin, probestin and bestatin

Harry H. Wasserman, Anders K. Petersen, Mingde Xia

Tetrahedron

Protease InhibitorsMedicinal ChemistryBiosynthesisBiochemistryNatural Sciences +10

Synthesis of the peptidic α-hydroxy amides phebestin, probestin, and bestatin from α-keto amide precursors

Harry H. Wasserman, Mingde Xia, Anders K. Petersen, +2

Tetrahedron Letters

Bioorganic ChemistryOrganic ChemistryPeptide ScienceChemical BiologyPharmaceutical Chemistry +16

Total Syntheses of Depsipeptide Elastase Inhibitors YM-47141 and YM-47142 with use of Ylide Protection and Coupling Methods

Harry H. Wasserman, Jyun‐Hung Chen, Mingde Xia

Journal of the American Chemical Society

Pharmaceutical ScienceDrug TargetBioorganic ChemistryAltmetric Attention ScorePeptide Science +16

A Sulfoxide-Based Ring Annelation Approach to Fused, Many-Membered Ring <b><i>N</i></b>,<b><i>S</i></b>-Heterocycles¹

Dallas K. Bates, Mingde Xia

The Journal of Organic Chemistry

Arylglycine derivatives as potent transient receptor potential melastatin 8 (TRPM8) antagonists

Bin Zhu, Mingde Xia, Xiaoqing Xu, +12

Bioorganic & Medicinal Chemistry Letters

Molecular PharmacologySignal TransductionBiochemistryFunctional SelectivityMedicine +8

Synthesis, Structure−Activity Relationship and in Vivo Antiinflammatory Efficacy of Substituted Dipiperidines as CCR2 Antagonists

Mingde Xia, Cuifen Hou, Duane E. DeMong, +11

Journal of Medicinal Chemistry

Pharmaceutical SciencePharmacotherapyChemistryChemical BiologyPharmaceutical Chemistry +16

Singlet oxygen oxidation of pyrroles. Formation of 5-substituted derivatives

Harry H. Wasserman, Mingde Xia, Jianji Wang, +2

Tetrahedron Letters

Tetrahydroindazole derivatives as potent and peripherally selective cannabinoid-1 (CB1) receptor inverse agonists

Jay M. Matthews, James J. McNally, Peter J. Connolly, +8

Bioorganic & Medicinal Chemistry Letters

Cannabis UsePsychoactive DrugTetrahydroindazole DerivativesSelective Cannabinoid-1Medicine +8

The Chemistry of Vicinal Tricarbonyls: Total Syntheses of Elastase Inhibitors YM-47141 and YM-47142

Harry H. Wasserman, Jyun‐Hung Chen, Mingde Xia

Helvetica Chimica Acta

First Natural ProductsBioorganic ChemistryPeptide ScienceElastase InhibitorsTotal Syntheses +15