Yuya Morita

Development of Orally Bioavailable Peptides Targeting an Intracellular Protein: From a Hit to a Clinical KRAS Inhibitor

Mikimasa Tanada, Minoru Tamiya, Atsushi Matsuo et al. · Journal of the American Chemical Society · 2023 · 132 citations

Chemoselective Boron-Catalyzed Nucleophilic Activation of Carboxylic Acids for Mannich-Type Reactions

Yuya Morita, Tomohiro Yamamoto, Hideoki Nagai et al. · Journal of the American Chemical Society · 2015 · 92 citations

Chemo- and Enantioselective Pd/B Hybrid Catalysis for the Construction of Acyclic Quaternary Carbons: Migratory Allylation of <i>O</i>-Allyl Esters to α-<i>C</i>-Allyl Carboxylic Acids

Taiki Fujita, Tomohiro Yamamoto, Yuya Morita et al. · Journal of the American Chemical Society · 2018 · 86 citations

Chemical Engineering, Cross-coupling Reaction, Engineering +15

Validation of a New Methodology to Create Oral Drugs beyond the Rule of 5 for Intracellular Tough Targets

Atsushi Ohta, Mikimasa Tanada, Shojiro Shinohara et al. · Journal of the American Chemical Society · 2023 · 86 citations

Data-driven catalyst optimization for stereodivergent asymmetric synthesis by iridium/boron hybrid catalysis

Hongyu Chen, Shigeru Yamaguchi, Yuya Morita et al. · Cell Reports Physical Science · 2021 · 50 citations · Full text