S. Malaquin

Ligand Efficiency Driven Design of New Inhibitors of <i>Mycobacterium tuberculosis</i> Transcriptional Repressor EthR Using Fragment Growing, Merging, and Linking Approaches

Baptiste Villemagne, Marion Flipo, Nicolas Blondiaux et al. · Journal of Medicinal Chemistry · 2014 · 64 citations · Full text

Medicinal Chemistry, Drug Target, Biochemistry +15

Ugi reaction for the synthesis of 4-aminopiperidine-4-carboxylic acid derivatives. Application to the synthesis of carfentanil and remifentanil

S. Malaquin, Mouhamad Jida, Jean‐Claude Gesquière et al. · Tetrahedron Letters · 2010 · 48 citations

Medicinal Chemistry, Natural Sciences, Ugi Reaction +9

Synthesis of five- and six-membered lactams via solvent-free microwave Ugi reaction

Mouhamad Jida, S. Malaquin, Rebecca Deprez‐Poulain et al. · Tetrahedron Letters · 2010 · 42 citations

Engineering, Organic Chemistry, Catalysis +5

Solvent-free microwave-assisted Meyers’ lactamization

Mouhamad Jida, Rebecca Deprez‐Poulain, S. Malaquin et al. · Green Chemistry · 2010 · 34 citations

Water-based conditions for the microscale parallel synthesis of bicyclic lactams

S. Malaquin, Mouhamad Jida, Justin Courtin et al. · Tetrahedron Letters · 2012 · 18 citations

Combinatorial Chemistry, Chemical Engineering, Engineering +8