A small molecule HIV-1 inhibitor that targets the HIV-1 envelope and inhibits CD4 receptor binding

Pin‐Fang Lin, Wade Blair, Tao Wang, +16

Proceedings of the National Academy of Sciences

ImmunologyMolecular BiologyImmunodominanceImmunotherapeuticsAntiviral Drug +17

BMS-232632, a Highly Potent Human Immunodeficiency Virus Protease Inhibitor That Can Be Used in Combination with Other Available Antiretroviral Agents

Brett S. Robinson, Keith Riccardi, Yi-Fei Gong, +8

Antimicrobial Agents and Chemotherapy

Biochemical and Genetic Characterizations of a Novel Human Immunodeficiency Virus Type 1 Inhibitor That Blocks gp120-CD4 Interactions

Qi Guo, Hsu‐Tso Ho, Ira B. Dicker, +14

Journal of Virology

ImmunologyMolecular BiologyBms-378806 BindsAntiviral DrugHuman Retrovirus +15

<i>In Vitro</i>Antiviral Characteristics of HIV-1 Attachment Inhibitor BMS-626529, the Active Component of the Prodrug BMS-663068

Beata Nowicka-Sans, Yi-Fei Gong, Brian McAuliffe, +18

Antimicrobial Agents and Chemotherapy

Prodrug Bms-663068Hiv-1 Gp120MedicineImmunologyAntiviral Response +11

Inhibitors of Human Immunodeficiency Virus Type 1 (HIV-1) Attachment. 5. An Evolution from Indole to Azaindoles Leading to the Discovery of 1-(4-Benzoylpiperazin-1-yl)-2-(4,7-dimethoxy-1<i>H</i>-pyrrolo[2,3-<i>c</i>]pyridin-3-yl)ethane-1,2-dione (BMS-488043), a Drug Candidate That Demonstrates Antiviral Activity in HIV-1-Infected Subjects

Tao Wang, Zhiwei Yin, Zhongxing Zhang, +23

Journal of Medicinal Chemistry

Organic ChemistryHiv-1-infected SubjectsPharmacotherapyAntiviral DrugAzaindole Leads +17

Niruriside, a New HIV REV/RRE Binding Inhibitor from <i>Phyllanthus niruri</i>

Jingfang Qian‐Cutrone, Stella Huang, John J. Trimble, +5

Journal of Natural Products

Specific Inhibitory ActivityMedicinal ChemistryBiochemistryBioassay-guided IsolationMedicine +10

Antiviral Activity, Pharmacokinetics, and Safety of BMS-488043, a Novel Oral Small-Molecule HIV-1 Attachment Inhibitor, in HIV-1-Infected Subjects

George J. Hanna, Jacob Lalezari, James Hellinger, +7

Antimicrobial Agents and Chemotherapy

High-resolution solution structure of siamycin II: Novel amphipathic character of a 21-residue peptide that inhibits HIV fusion

KeithL. Constantine, MarkS. Friedrichs, David J. Detlefsen, +9

Journal of Biomolecular NMR

Biochemistry21-Residue PeptideNatural SciencesMolecular BiologyPeptide Therapeutic +8

Assignment of the Murine Interferon Sensitivity and Cytoplasmic Superoxide Dismutase Genes to Chromosome 16

Pin‐Fang Lin, Doris L. Slate, Frances C. Lawyer, +1

Science

Knockout MouseChromatinPrimary Mouse CellsMurine Interferon SensitivityMouse Chromosome 16 +13

Initiation of genetic exchanges in λ phage-prophage crosses

Pin‐Fang Lin, Eva Bardwell, Paul Howard-Flanders

Proceedings of the National Academy of Sciences