<i>In Vitro</i>Antiviral Characteristics of HIV-1 Attachment Inhibitor BMS-626529, the Active Component of the Prodrug BMS-663068

Beata Nowicka-Sans, Yi-Fei Gong, Brian McAuliffe, +18

Antimicrobial Agents and Chemotherapy

Prodrug Bms-663068Hiv-1 Gp120MedicineImmunologyAntiviral Response +11

Envelope Conformational Changes Induced by Human Immunodeficiency Virus Type 1 Attachment Inhibitors Prevent CD4 Binding and Downstream Entry Events

Hsu‐Tso Ho, Fan Li, Beata Nowicka-Sans, +17

Journal of Virology

Antimicrobial Evaluation of Nocathiacins, a Thiazole Peptide Class of Antibiotics

Michael J. Pucci, Joanne J. Bronson, John F. Barrett, +4

Antimicrobial Agents and Chemotherapy

Bioorganic ChemistryAntimicrobial ChemotherapyL11 Ribosomal ProteinBacterial PathogensDrug Resistance +18

Novel water soluble phosphate prodrugs of taxol® possessing in vivo antitumor activity

Yasutsugu Ueda, Amarendra B. Mikkilineni, Jay O. Knipe, +3

Bioorganic & Medicinal Chemistry Letters

Medicinal ChemistryPharmaceutical ScienceTaxol® PossessingMedicinePolymer-drug Conjugate +7

Michael Addition of Amines and Thiols to Dehydroalanine Amides:  A Remarkable Rate Acceleration in Water

B. Narasimhulu Naidu, Margaret E. Sorenson, Timothy P. Connolly, +1

The Journal of Organic Chemistry

Derivative (Chemistry)Bioorganic ChemistryEngineeringBiochemistryNatural Sciences +11

Phosphonooxymethyl prodrugs of the broad spectrum antifungal azole, ravuconazole: Synthesis and biological properties

Yasutsugu Ueda, John D. Matiskella, Jerzy Golik, +19

Bioorganic & Medicinal Chemistry Letters

Antifungal AgentPhosphonooxymethyl ProdrugsBiochemistryAntifungal AgentsMedicine +6

Nocathiacin I analogues: synthesis, in vitro and in vivo biological activity of novel semi-synthetic thiazolyl peptide antibiotics

B. Narasimhulu Naidu, Margaret E. Sorenson, Yunhui Zhang, +10

Bioorganic & Medicinal Chemistry Letters

Medicinal ChemistryBiochemistryNatural SciencesMedicineVivo Biological Activity +5

Inhibitors of Human Immunodeficiency Virus Type 1 (HIV-1) Attachment 6. Preclinical and Human Pharmacokinetic Profiling of BMS-663749, a Phosphonooxymethyl Prodrug of the HIV-1 Attachment Inhibitor 2-(4-Benzoyl-1-piperazinyl)-1-(4,7-dimethoxy-1<i>H</i>-pyrrolo[2,3-<i>c</i>]pyridin-3-yl)-2-oxoethanone (BMS-488043)

John F. Kadow, Yasutsugu Ueda, Nicholas A. Meanwell, +15

Journal of Medicinal Chemistry

Synthesis, in vitro, and in vivo antibacterial activity of nocathiacin I thiol-Michael adducts

B. Narasimhulu Naidu, Margaret E. Sorenson, Joanne J. Bronson, +3

Bioorganic & Medicinal Chemistry Letters

Medicinal ChemistryMedicineAntibacterial AgentAntimicrobial ChemotherapyMicrobiology +4

Synthesis and evaluation of C2-carbon-linked heterocyclic-5-hydroxy-6-oxo-dihydropyrimidine-4-carboxamides as HIV-1 integrase inhibitors

B. Narasimhulu Naidu, Margaret E. Sorenson, Manoj Patel, +15

Bioorganic & Medicinal Chemistry Letters

EngineeringMedicineDrug DiscoveryAntiviral Drug DevelopmentOrganic Chemistry +6