Jia‐Ning Xiang

XP13512 [(±)-1-([(α-Isobutanoyloxyethoxy)carbonyl] aminomethyl)-1-cyclohexane Acetic Acid], A Novel Gabapentin Prodrug: I. Design, Synthesis, Enzymatic Conversion to Gabapentin, and Transport by Intestinal Solute Transporters

Kenneth C. Cundy, Russell Branch, Tania Chernov-Rogan et al. · Journal of Pharmacology and Experimental Therapeutics · 2004 · 151 citations

Pharmacy, Pharmacokinetics, Pharmacology +17

Development of an Enantioselective Synthetic Route to Neocarzinostatin Chromophore and Its Use for Multiple Radioisotopic Incorporation

Andrew G. Myers, Ralf Glatthar, Marlys Hammond et al. · Journal of the American Chemical Society · 2002 · 85 citations

Pharmacy, Chemistry, Medicinal Chemistry +10

Discovery of Biaryl Amides as Potent, Orally Bioavailable, and CNS Penetrant RORγt Inhibitors

Yonghui Wang, Wei Cai, Yaobang Cheng et al. · ACS Medicinal Chemistry Letters · 2015 · 76 citations · Full text

Pharmacy, Medicinal Chemistry, Pharmacology +10

Evaluation of Potent and Selective Small-Molecule Antagonists for the CXCR2 Chemokine Receptor

Katherine L. Widdowson, John D. Elliott, Daniel F. Veber et al. · Journal of Medicinal Chemistry · 2004 · 74 citations · Full text

Pharmacy, Medicinal Chemistry, Pharmacology +14

Discovery of novel N-(5-(arylcarbonyl)thiazol-2-yl)amides and N-(5-(arylcarbonyl)thiophen-2-yl)amides as potent RORγt inhibitors

Yonghui Wang, Wei Cai, Guifeng Zhang et al. · Bioorganic & Medicinal Chemistry · 2013 · 69 citations · Full text

Pharmacy, Medicinal Chemistry, Pharmacology +12