β₃-Adrenoceptor Is the Predominant β-Adrenoceptor Subtype in Human Myometrium and Its Expression Is Up-Regulated in Pregnancy

Céline Rouget, Marc Bardou, Michelle Breuiller-Fouché, +7

The Journal of Clinical Endocrinology & Metabolism

Identification of a novel snake peptide toxin displaying high affinity and antagonist behaviour for the α₂‐adrenoceptors

Céline Rouget, Loïc Quinton, Arhamatoulaye Maïga, +9

British Journal of Pharmacology

G protein-coupled receptors, an unexploited animal toxin targets: Exploration of green mamba venom for novel drug candidates active against adrenoceptors

Arhamatoulaye Maïga, Gilles Mourier, Loïc Quinton, +8

Toxicon

Signal TransductionBiochemistryG Protein-coupled ReceptorNovel Drug CandidatesGreen Mamba Venom +7

Modulation of nerve-evoked contractions by β3-adrenoceptor agonism in human and rat isolated urinary bladder

Céline Rouget, Moèz Rekik, Philippe Camparo, +5

Pharmacological Research

Adrenal GlandUrologyNeurophysiologyNerve-evoked ContractionsPhysiology +9

Nociceptin inhibits airway microvascular leakage induced by HCl intra‐oesophageal instillation

Céline Rouget, Yong Cui, Bruno D’Agostino, +4

British Journal of Pharmacology

The human near‐term myometrial <i>β</i>₃‐adrenoceptor but not the <i>β</i>₂‐adrenoceptor is resistant to desensitisation after sustained agonist stimulation

Céline Rouget, Michelle Breuiller-Fouché, F.J. Mercier, +8

British Journal of Pharmacology

Novel KV7 ion channel openers for the treatment of epilepsy and implications for detrusor tissue contraction

Mark A. Seefeld, Hong Lin, Joerg Holenz, +22

Bioorganic & Medicinal Chemistry Letters

Stimulation DeviceEngineeringHyperpolarization (Biology)NeurophysiologyPhysiology +6

In Vitro and in Vivo Pharmacological Characterization of Ethyl-4-{trans-4-[((2 S)-2-hydroxy-3-{4-hydroxy-3[(methylsulfonyl)amino]-phenoxy}propyl) Amino]cyclohexyl}benzoate Hydrochloride (SAR150640), a New Potent and Selective Human β3-Adrenoceptor Agonist for the Treatment of Preterm Labor

Tiziano Croci, Roberto Cecchi, Pietro Marini, +11

Journal of Pharmacology and Experimental Therapeutics

Involvement of β3-adrenoceptors in mouse urinary bladder function: Role in detrusor muscle relaxation and micturition reflex

Aurore Deba, Stéfano Palea, Céline Rouget, +2

European Journal of Pharmacology

UrologyVoiding DysfunctionMicturition ReflexMedicinePhysiology +5

Hypoxic Vasoconstriction of Rat Main Pulmonary Artery: Role of Endogenous Nitric Oxide, Potassium Channels, and Phosphodiesterase Inhibition

Marc Bardou, Françoise Goirand, Sandrine Marchand, +6

Journal of Cardiovascular Pharmacology

Pulmonary Arterial HypertensionPulmonary CirculationMedicineSelective PdeisPhysiology +13