New Folate-Grafted Chitosan Derivative To Improve Delivery of Paclitaxel-Loaded Solid Lipid Nanoparticles for Lung Tumor Therapy by Inhalation

Rémi Rosière, Matthias Van Woensel, Michel Gelbcke, +7

Molecular Pharmaceutics

NanoparticlesNanomedicineFolate ReceptorEngineeringPolymer-drug Conjugate +13

1-Synthesis of octa- and nonahelicenes. 2-New syntheses of hexa- and heptahelicenes. 3-Optical rotation and O.R.D. of heptahelicene.

R. H. Martin, M. Flammang‐Barbieux, J.P. Cosyn, +1

Tetrahedron Letters

EngineeringHeterocyclic2-New SynthesesOrganic Chemistry3-Optical Rotation +5

Structure–Activity Relationship Analysis of Bufadienolide-Induced in Vitro Growth Inhibitory Effects on Mouse and Human Cancer Cells

Laetitia Moreno Y Banuls, Ernst Urban, Michel Gelbcke, +4

Journal of Natural Products

Chemoprevention StrategyMouse Cancer CellsTumor BiologyMedicinal ChemistryCancer Cell Biology +17

Structure-Based Design, Synthesis, and Pharmacological Evaluation of 3-(Aminoalkyl)-5-fluoroindoles as Myeloperoxidase Inhibitors

Jalal Soubhye, Martine Prévost, Pierre Van Antwerpen, +9

Journal of Medicinal Chemistry

Combinatorial ChemistryLipid PeroxidationPeroxidase CyclesPharmacotherapyRedox Biology +19

Studies in NMR spectroscopy

R. H. Martin, N. Defay, H.P. Figeys, +4

Tetrahedron

Nmr SpectroscopyMagnetic Resonance SpectroscopySpectroscopyElectron Paramagnetic ResonanceResonance +5

Simple di- and trivanillates exhibit cytostatic properties toward cancer cells resistant to pro-apoptotic stimuli

Delphine Lamoral‐Theys, Laurent Pottier, Frédéric Kerff, +14

Bioorganic & Medicinal Chemistry

MedicineApoptosisCytostatic PropertiesMolecular BiologyAnti-cancer Agent +6

<i>N</i>-(2-{3-[3,5-Bis(trifluoromethyl)phenyl]ureido}ethyl)-glycyrrhetinamide (<b>6b</b>): A Novel Anticancer Glycyrrhetinic Acid Derivative that Targets the Proteasome and Displays Anti-Kinase Activity

Benjamin Lallemand, Fabien Chaix, Marina Bury, +10

Journal of Medicinal Chemistry

Discovery of Novel Potent Reversible and Irreversible Myeloperoxidase Inhibitors Using Virtual Screening Procedure

Jalal Soubhye, Ibaa Chikh Alard, Iyas Aldib, +14

Journal of Medicinal Chemistry

Drug TargetPharmacotherapyRedox BiologyPharmaceutical ChemistryStructure-based Virtual Screening +17

Design, Synthesis, and Structure–Activity Relationship Studies of Novel 3-Alkylindole Derivatives as Selective and Highly Potent Myeloperoxidase Inhibitors

Jalal Soubhye, Iyas Aldib, Betina Elfving, +16

Journal of Medicinal Chemistry

Pharmaceutical ScienceBioorganic ChemistryOrganic ChemistryFluoroindole CompoundChemical Biology +15

Interaction between dipyridamole and Eudragit S

D.B. Beten, Michel Gelbcke, B. Diallo, +1

International Journal of Pharmaceutics

Eudragit SChemistrySupramolecular Chemistry