M. J. MORCILLO

Optimization of the Pharmacophore Model for 5-HT₇R Antagonism. Design and Synthesis of New Naphtholactam and Naphthosultam Derivatives

María L. López-Rodrı́guez, Esther Porras, M. J. MORCILLO et al. · Journal of Medicinal Chemistry · 2003 · 70 citations · Full text

Synthesis and Structure−Activity Relationships of a New Model of Arylpiperazines. 2. Three-Dimensional Quantitative Structure−Activity Relationships of Hydantoin−Phenylpiperazine Derivatives with Affinity for 5-HT_1A and α₁ Receptors. A Comparison of CoMFA Models

María L. López-Rodrı́guez, M. Luisa Rosado, Bellinda Benhamú et al. · Journal of Medicinal Chemistry · 1997 · 64 citations · Full text

Synthesis and Structure−Activity Relationships of a New Model of Arylpiperazines. 1. 2-[[4-(<i>o</i>-Methoxyphenyl)piperazin-1-yl]methyl]-1,3- dioxoperhydroimidazo[1,5-<i>a</i>]pyridine:  A Selective 5-HT_1A Receptor Agonist

María L. López-Rodrı́guez, M. Luisa Rosado, Bellinda Benhamú et al. · Journal of Medicinal Chemistry · 1996 · 63 citations · Full text

Synthesis and Structure−Activity Relationships of a New Model of Arylpiperazines. 6. Study of the 5-HT_1A/α₁-Adrenergic Receptor Affinity by Classical Hansch Analysis, Artificial Neural Networks, and Computational Simulation of Ligand Recognition

María L. López-Rodrı́guez, M. J. MORCILLO, Esther Fernández et al. · Journal of Medicinal Chemistry · 2000 · 56 citations · Full text

Synthesis and Structure−Activity Relationships of a New Model of Arylpiperazines. 4. 1-[ω-(4-Arylpiperazin-1-yl)alkyl]-3-(diphenylmethylene)- 2,5-pyrrolidinediones and -3-(9<i>H</i>-fluoren-9-ylidene)-2,5-pyrrolidinediones: Study of the Steric Requirements of the Terminal Amide Fragment on 5-HT_1A Affinity/Selectivity

María L. López-Rodrı́guez, M. J. MORCILLO, Tandú K. Rovat et al. · Journal of Medicinal Chemistry · 1998 · 56 citations · Full text

Combinatorial Chemistry, Organic Chemistry, New Series +17