Alice Sebastian

14.beta.-[(p-Nitrocinnamoyl)amino]morphinones, 14.beta.-[(p-nitrocinnamoyl)amino]-7,8-dihydromorphinones, and their codeinone analogs: synthesis and receptor activity

Alice Sebastian, Jean M. Bidlack, Qing Jiang et al. · Journal of Medicinal Chemistry · 1993 · 29 citations · Full text

Asymmetric Syntheses, Opioid Receptor Affinities, and Antinociceptive Effects of 8-Amino-5,9-methanobenzocyclooctenes, a New Class of Structural Analogues of the Morphine Alkaloids

Arthur G. Schultz, Aihua Wang, Carlos Alva et al. · Journal of Medicinal Chemistry · 1996 · 23 citations · Full text

Nitrocinnamoyl and Chlorocinnamoyl Derivatives of Dihydrocodeinone: In Vivo and In Vitro Characterization of μ-Selective Agonist and Antagonist Activity

Jay P. McLaughlin, Kevin P. Hill, Qi Jiang et al. · Journal of Pharmacology and Experimental Therapeutics · 1999 · 16 citations

Development of a Pilot-Plant-Scale Synthesis of an Alkylated Dihydrobenzothiadiazole <i>S</i>,<i>S</i>-Dioxide: Incorporation of a Late-Stage Mitsunobu Reaction

Terrence J. Connolly, Waldemar P. Auguscinski, P. C. W. Fung et al. · Organic Process Research & Development · 2010 · 15 citations

Chemical Engineering, Diversity Oriented Synthesis, Engineering +13

14β-Chlorocinnamoylamino derivatives of metopon: long-term μ-opioid receptor antagonists

Jay P. McLaughlin, Alice Sebastian, Sydney Archer et al. · European Journal of Pharmacology · 1997 · 11 citations · Full text