Keizo Kan

Orally Active, Nonpeptide Vasopressin V₂ Receptor Antagonists:  A Novel Series of 1-[4-(Benzoylamino)benzoyl]-2,3,4,5-tetrahydro-1<i>H</i>-benzazepines and Related Compounds

Hidenori Ogawa, Hiroshi Yamashita, Kazumi Kondo et al. · Journal of Medicinal Chemistry · 1996 · 84 citations · Full text

Terminal Benzoyl Ring, Molecular Pharmacology, Medicinal Chemistry +13

Novel Design of Nonpeptide AVP V₂Receptor Agonists:  Structural Requirements for an Agonist Having 1-(4-Aminobenzoyl)-2,3,4,5-tetrahydro-1<i>H</i>-1-benzazepine as a Template

Kazumi Kondo, Hidenori Ogawa, Tomoichi Shinohara et al. · Journal of Medicinal Chemistry · 2000 · 62 citations · Full text

Po Administration, Novel Design, Pharmacotherapy +18

Characterization of Orally Active Nonpeptide Vasopressin V₂ Receptor Agonist. Synthesis and Biological Evaluation of Both the (5<i>R</i>)- and (5<i>S</i>)-Enantioisomers of 2-[1-(2-Chloro-4-pyrrolidin-1-yl-benzoyl)-2,3,4,5-tetrahydro-1<i>H</i>-1-benzazepin- 5-yl]-<i>N</i>-isopropylacetamide

Kazumi Kondo, Keizo Kan, Yoshihisa Tanada et al. · Journal of Medicinal Chemistry · 2002 · 45 citations · Full text

Pharmacotherapy, Experimental Pharmacology, Pharmaceutical Chemistry +17

Characterization of a novel nonpeptide vasopressin V₂‐agonist, OPC‐51803, in cells transfected human vasopressin receptor subtypes

Shigeki Nakamura, Yoshitaka Yamamura, S. Itoh et al. · British Journal of Pharmacology · 2000 · 30 citations · Full text

Immunology, Human Avp V, Pharmacotherapy +19

Investigation of the Carboxylate Position during the Acylation Reaction Catalyzed by Biaryl DMAP Derivatives with an Internal Carboxylate

Reiko Nishino, Takumi Furuta, Keizo Kan et al. · Angewandte Chemie International Edition · 2013 · 29 citations · Full text

Engineering, Carboxylate Position, Organic Chemistry +17