Concepedia

Eugene L. Piatnitski Chekler

EL

Statistics

Publications

22

Citations

1.2K

H-Index

15

Active since

2008

Affiliations

Pfizer (United States)(Current)

Merck KGaA, Darmstadt (Germany)

Ono Pharmaceutical (United States)

Eugene L. Piatnitski Chekler is an author at Pfizer (United States) specializing in medicinal chemistry, drug discovery, and pharmacy.

Publications per year

2008–2024

22

Publications

22

Target validation using chemical probes

Mark E. Bunnage, Eugene L. Piatnitski Chekler, Lyn H. Jones · Nature Chemical Biology · 2013 · 435 citations

, , +13

Large-Scale Assessment of Binding Free Energy Calculations in Active Drug Discovery Projects

Christina Schindler, Hannah M. Baumann, Andreas Blum et al. · Journal of Chemical Information and Modeling · 2020 · 311 citations

, , +14

Transcriptional Profiling of a Selective CREB Binding Protein Bromodomain Inhibitor Highlights Therapeutic Opportunities

Eugene L. Piatnitski Chekler, Jessica Pellegrino, Thomas A. Lanz et al. · Chemistry & Biology · 2015 · 60 citations · Full text

, , +8

Large-Scale Assessment of Binding Free Energy Calculations in Active Drug Discovery Projects

Christina Schindler, H Baumann, Andreas Blum et al. · ChemRxiv · 2020 · 51 citations · Full text

, , +14

Kiloscale Buchwald–Hartwig Amination: Optimized Coupling of Base-Sensitive 6-Bromoisoquinoline-1-carbonitrile with (<i>S</i>)-3-Amino-2-methylpropan-1-ol

Jeffrey B. Sperry, Kristin E. Price Wiglesworth, Ian D. Edmonds et al. · Organic Process Research & Development · 2014 · 45 citations

, , +13

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