Francesco Piscitelli

Arylthioindole Inhibitors of Tubulin Polymerization. 3. Biological Evaluation, Structure−Activity Relationships and Molecular Modeling Studies

Giuseppe La Regina, Michael Edler, Andrea Brancale et al. · Journal of Medicinal Chemistry · 2007 · 214 citations

Medicine, Medicinal Chemistry, Pharmacology +17

Design, Molecular Modeling, Synthesis, and Anti-HIV-1 Activity of New Indolyl Aryl Sulfones. Novel Derivatives of the Indole-2-carboxamide

Rino Ragno, Antonio Coluccia, Giuseppe La Regina et al. · Journal of Medicinal Chemistry · 2006 · 183 citations

Pharmacy, Medicinal Chemistry, Pharmacology +17

Toward Highly Potent Cancer Agents by Modulating the C-2 Group of the Arylthioindole Class of Tubulin Polymerization Inhibitors

Giuseppe La Regina, Ruoli Bai, Whilelmina Maria Rensen et al. · Journal of Medicinal Chemistry · 2012 · 124 citations · Full text

Medicine, Medicinal Chemistry, Pharmacology +13

New Arylthioindoles and Related Bioisosteres at the Sulfur Bridging Group. 4. Synthesis, Tubulin Polymerization, Cell Growth Inhibition, and Molecular Modeling Studies

Giuseppe La Regina, Taradas Sarkar, Ruoli Bai et al. · Journal of Medicinal Chemistry · 2009 · 88 citations · Full text

Pharmacy, Biochemistry, Medicinal Chemistry +15

Design and Synthesis of 2-Heterocyclyl-3-arylthio-1<i>H</i>-indoles as Potent Tubulin Polymerization and Cell Growth Inhibitors with Improved Metabolic Stability

Giuseppe La Regina, Ruoli Bai, Willeke Rensen et al. · Journal of Medicinal Chemistry · 2011 · 75 citations · Full text

Medicine, Medicinal Chemistry, Pharmacology +17