Sergey E. Tkachenko

Virtual and biomolecular screening converge on a selective agonist for GPR30

Cristian Bologa, Chetana M. Revankar, Susan Young et al. · Nature Chemical Biology · 2006 · 814 citations · Full text

Pharmacy, Medicinal Chemistry, Pharmacology +12

Synthesis and Structure–Activity Relationship (SAR) of (5,7-Disubstituted 3-phenylsulfonyl-pyrazolo[1,5-<i>a</i>]pyrimidin-2-yl)-methylamines as Potent Serotonin 5-HT₆Receptor (5-HT₆R) Antagonists

Alexandre V. Ivachtchenko, Elena S. Golovina, Volodymyr Kysil et al. · Journal of Medicinal Chemistry · 2011 · 106 citations · Full text

Medicine, Medicinal Chemistry, Pharmacology +17

Synthesis and Structure−Activity Relationship of 4-Substituted 2-(2-Acetyloxyethyl)-8-(morpholine- 4-sulfonyl)pyrrolo[3,4-<i>c</i>]quinoline- 1,3-diones as Potent Caspase-3 Inhibitors

Yulia A. Kuzovkova, Volodymyr Kysil, Sergey E. Tkachenko et al. · Journal of Medicinal Chemistry · 2005 · 84 citations · Full text

Pharmacy, Medicinal Chemistry, Pharmacology +13

Property-Based Design of GPCR-Targeted Library

Konstantin V. Balakin, Sergey E. Tkachenko, Stanley A. Lang et al. · Journal of Chemical Information and Computer Sciences · 2002 · 72 citations

Pharmacy, Medicinal Chemistry, Pharmacology +17

Pyrrolo[3,4-c]quinoline-1,3-diones as potent caspase-3 inhibitors. Synthesis and SAR of 2-substituted 4-methyl-8-(morpholine-4-sulfonyl)-pyrrolo[3,4-c]quinoline-1,3-diones

Volodymyr Kysil, Sergey E. Tkachenko, Sergey Maliarchouk et al. · European Journal of Medicinal Chemistry · 2005 · 64 citations

Pharmacy, Medicinal Chemistry, Pharmacology +9