Amol Gupte

5‘-<i>O</i>-[(<i>N</i>-Acyl)sulfamoyl]adenosines as Antitubercular Agents that Inhibit MbtA:  An Adenylation Enzyme Required for Siderophore Biosynthesis of the Mycobactins

Chunhua Qiao, Amol Gupte, Helena I. Boshoff et al. · Journal of Medicinal Chemistry · 2007 · 96 citations · Full text

Inhibition of Siderophore Biosynthesis by 2-Triazole Substituted Analogues of 5′-<i>O</i>-[<i>N</i>-(Salicyl)sulfamoyl]adenosine: Antibacterial Nucleosides Effective against <i>Mycobacterium tuberculosis</i>

Amol Gupte, Helena I. Boshoff, Daniel J. Wilson et al. · Journal of Medicinal Chemistry · 2008 · 84 citations · Full text

Synthesis and biological evaluation of isoxazole, oxazole, and oxadiazole containing heteroaryl analogs of biaryl ureas as DGAT1 inhibitors

Ravindra D. Jadhav, Kishorkumar S. Kadam, Shivaji Kandre et al. · European Journal of Medicinal Chemistry · 2012 · 50 citations · Full text

Medicinal Chemistry, Biochemistry, Biaryl Ureas +11

Copper(II)-Catalyzed Conversion of Aryl/Heteroaryl Boronic Acids, Boronates, and Trifluoroborates into the Corresponding Azides: Substrate Scope and Limitations

Courtney C. Aldrich, Kimberly D. Grimes, Amol Gupte · Synthesis · 2010 · 48 citations · Full text

Chemical Engineering, Cross-coupling Reaction, Engineering +13

Synthesis and biological evaluation of phloridzin analogs as human concentrative nucleoside transporter 3 (hCNT3) inhibitors

Amol Gupte, John K. Buolamwini · Bioorganic & Medicinal Chemistry Letters · 2008 · 33 citations · Full text

Molecular Pharmacology, Biochemistry, Medicine +7