K. Selvakumar

Discovery of an Oxycyclohexyl Acid Lysophosphatidic Acid Receptor 1 (LPA₁) Antagonist BMS-986278 for the Treatment of Pulmonary Fibrotic Diseases

Peter T. W. Cheng, Robert F. Kaltenbach, Hao Zhang et al. · Journal of Medicinal Chemistry · 2021 · 57 citations · Full text

Pharmacy, Medicinal Chemistry, Pharmacology +8

BMS-813160: A Potent CCR2 and CCR5 Dual Antagonist Selected as a Clinical Candidate

Robert J. Cherney, Prakash Anjanappa, K. Selvakumar et al. · ACS Medicinal Chemistry Letters · 2021 · 41 citations · Full text

Medicine, Pharmacokinetics, Pharmacology +14

Rationally Designed, Conformationally Constrained Inverse Agonists of RORγt—Identification of a Potent, Selective Series with Biologic-Like in Vivo Efficacy

David Marcoux, James J.‐W. Duan, Qing Shi et al. · Journal of Medicinal Chemistry · 2019 · 37 citations · Full text

Medicine, Medicinal Chemistry, Pharmacology +17

Discovery of a Hepatitis C Virus NS5B Replicase Palm Site Allosteric Inhibitor (BMS-929075) Advanced to Phase 1 Clinical Studies

Kap‐Sun Yeung, Brett R. Beno, Kyle Parcella et al. · Journal of Medicinal Chemistry · 2017 · 31 citations · Full text

Pharmacy, Medicinal Chemistry, Pharmacology +17

Electrophilicity of Pyridazine-3-carbonitrile, Pyrimidine-2-carbonitrile, and Pyridine-carbonitrile Derivatives: A Chemical Model To Describe the Formation of Thiazoline Derivatives in Human Liver Microsomes

Sarmistha Halder Sinha, Deepak Ahire, Santosh Wagh et al. · Chemical Research in Toxicology · 2014 · 21 citations

Life Sciences, Biochemistry, Pharmacology +14