Yannick J. Esvan

The <i>tert</i>-Butyl Side Chain: A Powerful Means to Lock Peptoid Amide Bonds in the Cis Conformation

Olivier Roy, Cécile Caumes, Yannick J. Esvan et al. · Organic Letters · 2013 · 102 citations · Full text

Life Sciences, Biochemistry, Supramolecular Chemistry +10

Discovery of pyrido[3,4-g]quinazoline derivatives as CMGC family protein kinase inhibitors: Design, synthesis, inhibitory potency and X-ray co–crystal structure

Yannick J. Esvan, Waël Zeinyeh, Thibaut Boibessot et al. · European Journal of Medicinal Chemistry · 2016 · 42 citations · Full text

Pharmacy, Chemistry, Medicinal Chemistry +16

New pyrido[3,4-g]quinazoline derivatives as CLK1 and DYRK1A inhibitors: synthesis, biological evaluation and binding mode analysis

Helmi Tazarki, Waël Zeinyeh, Yannick J. Esvan et al. · European Journal of Medicinal Chemistry · 2019 · 41 citations · Full text

Pharmacy, Medicinal Chemistry, Pharmacology +12

Synthesis and biological activity of pyrazole analogues of the staurosporine aglycon K252c

Yannick J. Esvan, F Giraud, Elisabeth Pereira et al. · Bioorganic & Medicinal Chemistry · 2016 · 20 citations · Full text

Pharmacy, Chemistry, Medicinal Chemistry +12

Regioselective cycloaddition of potassium alkynyltrifluoroborates with 3-azetidinones and 3-oxetanone by nickel-catalysed C–C bond activation

Fathi Elwrfalli, Yannick J. Esvan, Craig M. Robertson et al. · Chemical Communications · 2018 · 19 citations

Natural Sciences, Chemistry, Medicinal Chemistry +15