Concepedia
Author
Sigrid Hatse
Also Known As
Anne-Sophie Dieudonne, Caroline Weltens, Hatse, Sigrid, S Hatse, S. Hatse, Shu, X.-O., Sigrid Hatse, Sigrid Hatse (12560)
205
Publications
5.9K
Citations
42
H-Index
92
Concepts
All Affiliations
1
20
23
2.3K
2
4
587
3
551
179
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All Concepts
66
4.5K
37
Multidrug-resistance protein 5 is a multispecific organic anion transporter able to transport nucleotide analogs
Jan Wijnholds, Carla A.A.M. Mol, Liesbeth van Deemter, +9
Proceedings of the National Academy of Sciences
Molecular PharmacologyHuman Mrp5Proteinlipid InteractionMultidrug-resistance Protein 5Biochemistry +13
2000
472
Chemokine receptor inhibition by AMD3100 is strictly confined to CXCR4
Sigrid Hatse, Katrien Princen, Gary Bridger, +2
FEBS Letters
InflammationCytokineCxcr4 InternalizationSignal TransductionMedicine +13
2002
446
AMD3100, a Potent and Specific Antagonist of the Stromal Cell-Derived Factor-1 Chemokine Receptor CXCR4, Inhibits Autoimmune Joint Inflammation in IFN-γ Receptor-Deficient Mice
Patrick Matthys, Sigrid Hatse, Kurt Vermeire, +6
The Journal of Immunology
Specific AntagonistImmunologyImmune RegulationCd4 T Cell ResponsesInnate Immunity +19
2001
Mannose-Specific Plant Lectins from the <i>Amaryllidaceae</i> Family Qualify as Efficient Microbicides for Prevention of Human Immunodeficiency Virus Infection
Jan Balzarini, Sigrid Hatse, Kurt Vermeire, +9
Antimicrobial Agents and Chemotherapy
2004
147
A palmitate-rich metastatic niche enables metastasis growth via p65 acetylation resulting in pro-metastatic NF-κB signaling
Patricia Altea‐Manzano, Ginevra Doglioni, Yawen Liu, +47
Nature Cancer
P65 AcetylationPro-metastatic Nf-κb SignalingSignaling PathwayMedicineRadiation Oncology +7
2023
128
AMD3465, a monomacrocyclic CXCR4 antagonist and potent HIV entry inhibitor
Sigrid Hatse, Katrien Princen, Erik De Clercq, +6
Biochemical Pharmacology
Human RetrovirusPharmacologyImmunologyAntiviral ResponseAntiviral Drug Development +7
2005
123
Carbohydrate-binding Agents Cause Deletions of Highly Conserved Glycosylation Sites in HIV GP120
Jan Balzarini, Kristel Van Laethem, Sigrid Hatse, +4
Journal of Biological Chemistry
Discovery of Novel Small Molecule Orally Bioavailable C−X−C Chemokine Receptor 4 Antagonists That Are Potent Inhibitors of T-Tropic (X4) HIV-1 Replication
Renato T. Skerlj, Gary Bridger, Al Kaller, +13
Journal of Medicinal Chemistry
2010
115
Mutation of Asp<sup>171</sup>and Asp<sup>262</sup>of the Chemokine Receptor CXCR4 Impairs Its Coreceptor Function for Human Immunodeficiency Virus-1 Entry and Abrogates the Antagonistic Activity of AMD3100
Sigrid Hatse, Katrien Princen, Lars‐Ole Gerlach, +5
Molecular Pharmacology
113
Molecular Mechanism of Action of Monocyclam Versus Bicyclam Non-peptide Antagonists in the CXCR4 Chemokine Receptor
Mette M. Rosenkilde, Lars-Ole Gerlach, Sigrid Hatse, +4
2007
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