Shoichi Sagawa

Catalytic Asymmetric Aminolysis of 3,5,8-Trioxabicyclo[5.1.0]octane Providing an Optically Pure 2-Amino-1,3,4-butanetriol Equivalent

Shoichi Sagawa, Hiroyuki Abé, Yasunori Hase et al. · The Journal of Organic Chemistry · 1999 · 139 citations

Catalytic Asymmetric Aminolysis, Engineering, Heterocyclic +13

Synthesis of anilino-monoindolylmaleimides as potent and selective PKCβ inhibitors

Masahiro Tanaka, Shoichi Sagawa, Jun‐ichi Hoshi et al. · Bioorganic & Medicinal Chemistry Letters · 2004 · 61 citations · Full text

Medicine, Selective Pkcβ Inhibitors, Pharmacology +2

(1<i>S</i>)-1-[(4<i>R</i>)-2,2-Dimethyl-1,3-dioxolan-4-yl]-2-hydroxyethylammonium Benzoate, A Versatile Building Block for Chiral 2-Aminoalkanols:  Concise Synthesis and Application to Nelfinavir, a Potent HIV-Protease Inhibitor

Takashi Inaba, Yasuki Yamada, Hiroyuki Abé et al. · The Journal of Organic Chemistry · 2000 · 48 citations

Bioorganic Chemistry, Organic Chemistry, Antiviral Drug +17

Synthesis, SAR studies, and pharmacological evaluation of 3-anilino-4-(3-indolyl) maleimides with conformationally restricted structure as orally bioavailable PKCβ-selective inhibitors

Masahiro Tanaka, Shoichi Sagawa, Jun‐ichi Hoshi et al. · Bioorganic & Medicinal Chemistry · 2006 · 44 citations

Pharmaceutical Science, Biochemistry, Medicine +9

Novel protein kinase C‐β isoform selective inhibitor JTT‐010 ameliorates both hyper‐ and hypoalgesia in streptozotocin‐ induced diabetic rats

Tomohiko Sasase, Hideki Yamada, Kenji Sakoda et al. · Diabetes Obesity and Metabolism · 2004 · 42 citations