Thierry Drujon

Synthesis and Evaluation of Analogues of <i>N</i>-Phthaloyl-<scp>l</scp>-tryptophan (RG108) as Inhibitors of DNA Methyltransferase 1

Saâdia Asgatay, Christine Champion, Gaël Marloie et al. · Journal of Medicinal Chemistry · 2013 · 95 citations · Full text

Combinatorial Chemistry, Molecular Biology, Organic Chemistry +17

Rapid Synthesis of New DNMT Inhibitors Derivatives of Procainamide

Ludovic Halby, Christine Champion, Catherine Sénamaud‐Beaufort et al. · ChemBioChem · 2011 · 61 citations

Label-free measurement of histone lysine methyltransferases activity by matrix-assisted laser desorption/ionization time-of-flight mass spectrometry

Karine Guitot, Silvia Scarabelli, Thierry Drujon et al. · Analytical Biochemistry · 2014 · 21 citations

Label-free Measurement, Biochemistry, Analytical Instrumentation +11

A direct label-free MALDI-TOF mass spectrometry based assay for the characterization of inhibitors of protein lysine methyltransferases

Karine Guitot, Thierry Drujon, Fabienne Burlina et al. · Analytical and Bioanalytical Chemistry · 2017 · 21 citations

Molecular Characterization, Biochemistry, Medicine +10

Inhibition of Diamino Pelargonic Acid Aminotransferase, an Enzyme of the Biotin Biosynthetic Pathway, by Amiclenomycin: A Mechanistic Study

Stéphane Mann, Dominique Florentin, Denis Lesage et al. · Helvetica Chimica Acta · 2003 · 15 citations

Peptide Science, Mechanistic Study, Biotin Biosynthetic Pathway +21