The Interaction of Charged and Uncharged Drugs with Neutral (HP-β-CD) and Anionically Charged (SBE7-β-CD) β-Cyclodextrins

Kazuto Okimoto, Roger A. Rajewski, Kaneto Uekama, +2

Pharmaceutical Research

Fast Surface Crystallization of Amorphous Griseofulvin Below T g

Lei Zhu, Janan Jona, Karthik Nagapudi, +1

Pharmaceutical Research

Materials ScienceEngineeringCrystal Growth TechnologySurface ScienceApplied Physics +3

A Quantitative Kinetic Study of Polysorbate Autoxidation: The Role of Unsaturated Fatty Acid Ester Substituents

Yao Jia, Dushyanth K. Dokuru, Matthew Noestheden, +5

Pharmaceutical Research

Food ChemistryLipid AnalysisBiochemistryOmega-3 Fatty AcidPolysorbate Autoxidation +2

Discovery of a Potent, Orally Active 11β-Hydroxysteroid Dehydrogenase Type 1 Inhibitor for Clinical Study: Identification of (<i>S</i>)-2-((1<i>S</i>,2<i>S</i>,4<i>R</i>)-Bicyclo[2.2.1]heptan-2-ylamino)-5-isopropyl-5-methylthiazol-4(5<i>H</i>)-one (AMG 221)

Murielle M. Véniant, Clarence Hale, Randall W. Hungate, +23

Journal of Medicinal Chemistry

Molecular PharmacologyMedicinal ChemistryMethyl GroupBiochemistryC-5 Position +12

High‐throughput logP measurement using parallel liquid chromatography/ultraviolet/mass spectrometry and sample‐pooling

Yining Zhao, Janan Jona, David Chow, +6

Rapid Communications in Mass Spectrometry

Lead CompoundsEngineeringChemistryHigh-throughput Logp MeasurementEnvironmental Chemistry +16

Amorphous Active Pharmaceutical Ingredients in Preclinical Studies: Preparation, Characterization, and Formulation

Karthik Nagapudi, Janan Jona

Current Bioactive Compounds

Pharmaceutical ScienceChemistryPharmaceutical ChemistrySolution (Chemistry)Pharmaceutical Formulation +14

Manufacture and Performance Evaluation of a Stable Amorphous Complex of an Acidic Drug Molecule and Neusilin

Jenifer Anne MacLean, César Medina, Dominick Daurio, +4

Journal of Pharmaceutical Sciences

Combinatorial ChemistryMedicinal ChemistryPharmaceutical ScienceNatural SciencesAcidic Drug Molecule +7

Applications of modulated differential scanning calorimetry in preformulation studies

Shelley R. Rabel, Janan Jona, Michael B. Maurin

Journal of Pharmaceutical and Biomedical Analysis

EngineeringDifferential Scanning CalorimetryMeasurementCalibrationEducation +7

Preparation of 1-(3-aminobenzo[d]isoxazol-5-yl)-1H-pyrazolo[4,3-d]pyrimidin-7(6H)-ones as potent, selective, and efficacious inhibitors of coagulation factor Xa

Yunlong Li, John M. Fevig, Joseph Cacciola, +9

Bioorganic & Medicinal Chemistry Letters

Medicinal ChemistryPharmaceutical ScienceBiochemistryAntiparasitic AgentMedicine +9

Quantitative determination of solid-state forms of a pharmaceutical development compound in drug substance and tablets

Yong Xie, Wenle Tao, Henry Morrison, +4

International Journal of Pharmaceutics

Drug SubstanceChemical MeasurementMedicineDrug PurityQuantitative Determination +9