Jeffrey B. Arterburn

A Transmembrane Intracellular Estrogen Receptor Mediates Rapid Cell Signaling

Chetana M. Revankar, Daniel F. Cimino, Larry A. Sklar et al. · Science · 2005 · 2.3K citations

Virtual and biomolecular screening converge on a selective agonist for GPR30

Cristian Bologa, Chetana M. Revankar, Susan Young et al. · Nature Chemical Biology · 2006 · 805 citations · Full text

Drug Target, G Protein-coupled Receptor, Medicine +9

In vivo effects of a GPR30 antagonist

Megan K. Dennis, Ritwik Burai, Chinnasamy Ramesh et al. · Nature Chemical Biology · 2009 · 514 citations · Full text

Functional Selectivity, Medicine, Pharmacological Agent +5

Identification of a GPER/GPR30 antagonist with improved estrogen receptor counterselectivity

Megan K. Dennis, Angela S. Field, Ritwik Burai et al. · The Journal of Steroid Biochemistry and Molecular Biology · 2011 · 303 citations · Full text

Endocrine Mechanism, Gper/gpr30 Antagonist, Medicine +7

GPR30 Expression Is Required for the Mineralocorticoid Receptor–Independent Rapid Vascular Effects of Aldosterone

Robert Gros, Qingming Ding, Larry A. Sklar et al. · Hypertension · 2011 · 238 citations · Full text

Molecular Pharmacology, Endocrine Mechanism, Medicine +13