Michel Enderlin-Paput

Design, Synthesis, and Characterization of Novel Tetrahydropyran-Based Bacterial Topoisomerase Inhibitors with Potent Anti-Gram-Positive Activity

Jean‐Philippe Surivet, Cornelia Zumbrunn, Georg Rueedi et al. · Journal of Medicinal Chemistry · 2013 · 67 citations · Full text

Life Sciences, Medicinal Chemistry, Pharmacology +17

Discovery of Novel Inhibitors of LpxC Displaying Potent in Vitro Activity against Gram-Negative Bacteria

Jean‐Philippe Surivet, Philippe Panchaud, Jean‐Luc Specklin et al. · Journal of Medicinal Chemistry · 2019 · 37 citations

Pharmacy, Medicinal Chemistry, Pharmacology +17

Synthesis and Characterization of Tetrahydropyran-Based Bacterial Topoisomerase Inhibitors with Antibacterial Activity against Gram-Negative Bacteria

Jean‐Philippe Surivet, Cornelia Zumbrunn, Thierry Bruyère et al. · Journal of Medicinal Chemistry · 2017 · 35 citations · Full text

Pharmacy, Medicinal Chemistry, Pharmacology +17

Novel Tetrahydropyran-Based Bacterial Topoisomerase Inhibitors with Potent Anti-Gram Positive Activity and Improved Safety Profile

Jean‐Philippe Surivet, Cornelia Zumbrunn, Georg Rueedi et al. · Journal of Medicinal Chemistry · 2014 · 33 citations

Pharmacy, Medicinal Chemistry, Pharmacology +17

Optimization of LpxC Inhibitor Lead Compounds Focusing on Efficacy and Formulation for High Dose Intravenous Administration

Philippe Panchaud, Jean‐Philippe Surivet, Stefan Diethelm et al. · Journal of Medicinal Chemistry · 2019 · 17 citations · Full text

Pharmacy, Medicinal Chemistry, Pharmacology +17