Concepedia
Statistics
Publications
7
Citations
480
H-Index
Active since
1998
Affiliations
Bial (Portugal)(Current)
Eötvös Loránd University
Universidade do Porto
László E. Kiss is an author at Bial (Portugal) specializing in medicine, drug discovery, and natural sciences.
Top concepts
MedicineDrug DiscoveryPharmacologyNatural SciencesMedicinal ChemistryChemistryBiochemistryPharmacotherapyDrug DevelopmentOrganic Chemistry
Publications per year
1998–2018
Discovery of a Long-Acting, Peripherally Selective Inhibitor of Catechol-<i>O</i>-methyltransferase
László E. Kiss, Humberto Ferreira, Leonel Torrão et al. · Journal of Medicinal Chemistry · 2010 · 164 citations
Bioorganic Chemistry, Pharmacotherapy, Chemical Biology +16
An improved design of fluorophilic molecules: prediction of the ln P fluorous partition coefficient, fluorophilicity, using 3D QSAR descriptors and neural networks
László E. Kiss, István Kövesdi, József Rábai · Journal of Fluorine Chemistry · 2001 · 102 citations
Engineering, Fluorophilic Molecules, Improved Design +11
Medicinal Chemistry of Catechol<i>O</i>-Methyltransferase (COMT) Inhibitors and Their Therapeutic Utility
László E. Kiss, Patrício Soares‐da‐Silva · Journal of Medicinal Chemistry · 2014 · 100 citations
Medicinal Chemistry, Pharmaceutical Science, Biochemistry +13
Efficient Synthesis of 2-(Trifluoromethyl)nicotinic Acid Derivatives from Simple Fluorinated Precursors
László E. Kiss, Humberto Ferreira, David A. Learmonth · Organic Letters · 2008 · 47 citations
Nicotinic Acid Derivatives, Organic Chemistry, Chemistry +16
Design, synthesis, and structure–activity relationships of 1,3,4-oxadiazol-2(3H)-ones as novel FAAH inhibitors
László E. Kiss, Humberto Ferreira, Leonel Torrão et al. · MedChemComm · 2011 · 26 citations
Medicinal Chemistry, Pharmaceutical Science, Biochemistry +15
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