Edelweiss Evrard

Introduction of a Crystalline, Shelf-Stable Reagent for the Synthesis of Sulfur(VI) Fluorides

Hua Zhou, Paramita Mukherjee, Rongqiang Liu et al. · Organic Letters · 2018 · 140 citations

Natural Sciences, Chemical Engineering, Chemistry +8

Discovery of Brain-Penetrant, Irreversible Kynurenine Aminotransferase II Inhibitors for Schizophrenia

Amy B. Dounay, Marie Anderson, Bruce M. Bechle et al. · ACS Medicinal Chemistry Letters · 2012 · 90 citations · Full text

Pharmacy, Medicinal Chemistry, Pharmacology +13

Discovery of 4-(5-Methyloxazolo[4,5-<i>b</i>]pyridin-2-yl)-1,4-diazabicyclo[3.2.2]nonane (CP-810,123), a Novel α7 Nicotinic Acetylcholine Receptor Agonist for the Treatment of Cognitive Disorders in Schizophrenia: Synthesis, SAR Development, and in Vivo Efficacy in Cognition Models

Christopher J. O’Donnell, Bruce N. Rogers, Brian S. Bronk et al. · Journal of Medicinal Chemistry · 2009 · 74 citations · Full text

Pharmacy, Pharmacology, Pharmacotherapy +17

PF-04859989 as a template for structure-based drug design: Identification of new pyrazole series of irreversible KAT II inhibitors with improved lipophilic efficiency

Amy B. Dounay, Marie Anderson, Bruce M. Bechle et al. · Bioorganic & Medicinal Chemistry Letters · 2013 · 32 citations · Full text

Pharmacy, Medicinal Chemistry, Pharmacology +16

Photoaffinity Labeling and Quantitative Chemical Proteomics Identify LXRβ as the Functional Target of Enhancers of Astrocytic apoE

Uthpala Seneviratne, Zhen Huang, Christopher W. am Ende et al. · Cell chemical biology · 2020 · 27 citations

Life Sciences, Biochemistry, Molecular Biology +14