Eyad K. Fansa

Identification of pyrazolopyridazinones as PDEδ inhibitors

Bjoern Papke, Sandip Murarka, Holger A. Vogel et al. · Nature Communications · 2016 · 162 citations · Full text

Medicine, Oncology, Pharmacology +12

Activating mutations in RRAS underlie a phenotype within the RASopathy spectrum and contribute to leukaemogenesis

Elisabetta Flex, Mamta Jaiswal, Francesca Pantaleoni et al. · Human Molecular Genetics · 2014 · 142 citations · Full text

Medicine, Genetics, Molecular Genetics +17

Covalent Protein Labeling at Glutamic Acids

Pablo Martín‐Gago, Eyad K. Fansa, Michael Winzker et al. · Cell chemical biology · 2017 · 97 citations · Full text

Life Sciences, Biochemistry, Molecular Biology +14

A PDE6δ‐KRas Inhibitor Chemotype with up to Seven H‐Bonds and Picomolar Affinity that Prevents Efficient Inhibitor Release by Arl2

Pablo Martín‐Gago, Eyad K. Fansa, Christian H. Klein et al. · Angewandte Chemie International Edition · 2017 · 88 citations

Medicine, Medicinal Chemistry, Pharmacology +15

PDE6δ-mediated sorting of INPP5E into the cilium is determined by cargo-carrier affinity

Eyad K. Fansa, Stefanie Kristine Kösling, Eldar Zent et al. · Nature Communications · 2016 · 85 citations · Full text

Life Sciences, Cell Biology, Molecular Biology +17