Gaoqiang Yang

New Angiopep-Modified Doxorubicin (ANG1007) and Etoposide (ANG1009) Chemotherapeutics With Increased Brain Penetration

Christian Ché, Gaoqiang Yang, Carine Thiot et al. · Journal of Medicinal Chemistry · 2010 · 130 citations

Immunology, Brain Penetration, Cell Death +22

Structure-Based Design, Synthesis, and Memapsin 2 (BACE) Inhibitory Activity of Carbocyclic and Heterocyclic Peptidomimetics

Stephen Hanessian, Hongying Yun, Yihua Hou et al. · Journal of Medicinal Chemistry · 2005 · 72 citations · Full text

Combinatorial Chemistry, Medicinal Chemistry, Biochemistry +13

Structure-Based Design and Synthesis of Macroheterocyclic Peptidomimetic Inhibitors of the Aspartic Protease β-Site Amyloid Precursor Protein Cleaving Enzyme (BACE)

Stephen Hanessian, Gaoqiang Yang, Jean‐Michel Rondeau et al. · Journal of Medicinal Chemistry · 2006 · 61 citations · Full text

Synthesis of enantiomerically pure α-amino-β-hydroxy-cyclobutanone derivatives and their transformations into polyfunctional three- and five-membered ring compounds

Léon Ghosez, Gaoqiang Yang, José Renato Cagnon et al. · Tetrahedron · 2004 · 26 citations

Derivatives, Biochemistry, Organic Chemistry +5

Use of a Noninvasive Brain-Penetrating Peptide-Drug Conjugate Strategy to Improve the Delivery of Opioid Pain Relief Medications to the Brain

E Eiselt, Valérie Otis, Karine Belleville et al. · Journal of Pharmacology and Experimental Therapeutics · 2020 · 17 citations · Full text