Andrew S. Thompson

Direct conversion of activated alcohols to azides using diphenyl phosphorazidate. A practical alternative to Mitsunobu conditions

Andrew S. Thompson, Guy R. Humphrey, A. M. DEMARCO et al. · The Journal of Organic Chemistry · 1993 · 303 citations

Natural Sciences, Chemistry, Analytical Chemistry +4

Practical Asymmetric Synthesis of Efavirenz (DMP 266), an HIV-1 Reverse Transcriptase Inhibitor

Michael E. Pierce, Rodney L. Parsons, Lilian Radesca et al. · The Journal of Organic Chemistry · 1998 · 215 citations

Pharmacy, Chemistry, Medicinal Chemistry +16

Lithium Ephedrate-Mediated Addition of a Lithium Acetylide to a Ketone:  Solution Structures and Relative Reactivities of Mixed Aggregates Underlying the High Enantioselectivities

Andrew S. Thompson, Edward G. Corley, Martha Huntington et al. · Journal of the American Chemical Society · 1998 · 162 citations

Natural Sciences, Chemistry, Catalysis +10

Rational design of a highly efficient irreversible DNA interstrand cross-linking agent based on the pyrrolobenzodiazepine ring system

D. Subhas Bose, Andrew S. Thompson, Jingshan Ching et al. · Journal of the American Chemical Society · 1992 · 136 citations

Pharmacy, Medicinal Chemistry, Bioorthogonal Chemistry +8

Use of an ephedrine alkoxide to mediate enantioselective addition of an acetylide to a prochiral ketone: asymmetric synthesis of the reverse transcriptase inhibitor L-743,726

Andrew S. Thompson, Edward G. Corley, Martha Huntington et al. · Tetrahedron Letters · 1995 · 131 citations

Natural Sciences, Chemistry, Medicinal Chemistry +13