Charles W. Lugar

Structure−Activity Relationships of Selective Estrogen Receptor Modulators:  Modifications to the 2-Arylbenzothiophene Core of Raloxifene

Timothy A. Grese, Stephen Cho, Don R. Finley et al. · Journal of Medicinal Chemistry · 1997 · 175 citations · Full text

Gynecology, Raloxifene Analogs, Pharmacotherapy +23

Benzopyrans Are Selective Estrogen Receptor β Agonists with Novel Activity in Models of Benign Prostatic Hyperplasia

Bryan H. Norman, Jeffrey A. Dodge, Timothy I. Richardson et al. · Journal of Medicinal Chemistry · 2006 · 102 citations · Full text

Gynecology, Pharmacotherapy, Novel Activity +16

Evaluation of the major metabolites of raloxifene as modulators of tissue selectivity

Jeffrey A. Dodge, Charles W. Lugar, Stephen Cho et al. · The Journal of Steroid Biochemistry and Molecular Biology · 1997 · 55 citations

Medicinal Chemistry, Pharmacological Study, Biochemistry +9

Novel 3-Aryl Indoles as Progesterone Receptor Antagonists for Uterine Fibroids

Timothy I. Richardson, Christian A. Clarke, Kuo‐Long Yu et al. · ACS Medicinal Chemistry Letters · 2010 · 50 citations · Full text

Medicinal Chemistry, Hormonal Contraceptive, Uterine Fibroids +15

Structure−Activity Studies of 6-(Tetrazolylalkyl)-Substituted Decahydroisoquinoline-3-carboxylic Acid AMPA Receptor Antagonists. 1. Effects of Stereochemistry, Chain Length, and Chain Substitution

Paul L. Ornstein, M. Brian Arnold, Nancy K. Allen et al. · Journal of Medicinal Chemistry · 1996 · 47 citations