Alessandro Ettorre

Structure-Based Design, Synthesis, and Biological Evaluation of Novel Pyrrolyl Aryl Sulfones:  HIV-1 Non-Nucleoside Reverse Transcriptase Inhibitors Active at Nanomolar Concentrations

Marino Artico, Romano Silvestri, E. PAGNOZZI et al. · Journal of Medicinal Chemistry · 2000 · 133 citations · Full text

Configurational requirements of the sugar moiety for the pharmacological activity of anthracycline disaccharides

Federico Arcamone, Fabio Animati, Mario Bigioni et al. · Biochemical Pharmacology · 1999 · 34 citations

Bioorganic Chemistry, Glycosylation, Biochemistry +10

hNK2 receptor antagonists. The use of intramolecular hydrogen bonding to increase solubility and membrane permeability

Alessandro Ettorre, Piero D’Andrea, Sandro Mauro et al. · Bioorganic & Medicinal Chemistry Letters · 2011 · 33 citations · Full text

Molecular Pharmacology, Intramolecular Hydrogen, Hnk2 Receptor Antagonists +10

Conformational restriction through Cαi ←→ Cαi cyclization: 1-aminocycloheptane-1-carboxylic acid (Ac7c)

Ettore Benedetti, Benedetto Di Blasio, Rosa Iacovino et al. · Journal of the Chemical Society Perkin Transactions 2 · 1997 · 26 citations

Engineering, Conformational Restriction, Biochemistry +12

Alkyl piperidine and piperazine hydroxamic acids as HDAC inhibitors

Cristina Rossi, Marina Porcelloni, Piero D’Andrea et al. · Bioorganic & Medicinal Chemistry Letters · 2011 · 23 citations · Full text

Molecular Pharmacology, Medicinal Chemistry, Hdac Inhibitors +7