Katharine Grant-Young

4-Thiazolidinones: novel inhibitors of the bacterial enzyme murB

Charles J. Andres, Joanne J. Bronson, Stanley V. D’Andrea et al. · Bioorganic & Medicinal Chemistry Letters · 2000 · 220 citations

Life Sciences, Medicinal Chemistry, Microbiology +9

Discovery and Preclinical Characterization of the Cyclopropylindolobenzazepine BMS-791325, A Potent Allosteric Inhibitor of the Hepatitis C Virus NS5B Polymerase

Robert G. Gentles, Min Ding, John A. Bender et al. · Journal of Medicinal Chemistry · 2014 · 100 citations · Full text

Pharmacy, Medicinal Chemistry, Pharmacology +17

Structure–activity relationships for a series of thiobenzamide influenza fusion inhibitors derived from 1,3,3-Trimethyl-5-hydroxy-cyclohexylmethylamine

Kuo-Long Yu, Albert Torri, Guangxiang Luo et al. · Bioorganic & Medicinal Chemistry Letters · 2002 · 51 citations

Pharmacy, Medicinal Chemistry, Pharmacology +13

Identification of a Potent and Selective 5-HT₆Antagonist:  One-Step Synthesis of (<i>E</i>)-3-(Benzenesulfonyl)-2- (methylsulfanyl)pyrido[1,2-<i>a</i>]pyrimidin- 4-ylidenamine from 2-(Benzenesulfonyl)-3,3- bis(methylsulfanyl)acrylonitrile

Yong‐Jin Wu, Huan He, Shuanghua Hu et al. · Journal of Medicinal Chemistry · 2003 · 28 citations · Full text

Pharmacy, Medicinal Chemistry, Pharmacology +9

Improving Metabolic Stability with Deuterium: The Discovery of BMT-052, a Pan-genotypic HCV NS5B Polymerase Inhibitor

Kyle Parcella, Kyle J. Eastman, Kap‐Sun Yeung et al. · ACS Medicinal Chemistry Letters · 2017 · 26 citations · Full text

Pharmacy, Medicinal Chemistry, Pharmacology +13