Mickaël Maudet

Discovery of (<i>R</i>)-8-(1-(3,5-Difluorophenylamino)ethyl)-<i>N</i>,<i>N</i>-dimethyl-2-morpholino-4-oxo-4<i>H</i>-chromene-6-carboxamide (AZD8186): A Potent and Selective Inhibitor of PI3Kβ and PI3Kδ for the Treatment of PTEN-Deficient Cancers

Bernard Barlaam, Sabina Cosulich, Sébastien L. Degorce et al. · Journal of Medicinal Chemistry · 2014 · 85 citations · Full text

Pten Deficient Tumors, Pharmacotherapy, Pharmaceutical Chemistry +20

Investigation of (<i>E</i>)-3-[4-(2-Oxo-3-aryl-chromen-4-yl)oxyphenyl]acrylic Acids as Oral Selective Estrogen Receptor Down-Regulators

Sébastien L. Degorce, Andrew Bailey, Rowena Callis et al. · Journal of Medicinal Chemistry · 2015 · 42 citations · Full text

Breast Oncology, Female Reproductive Function, Pharmacotherapy +19

Asymmetric synthesis of (S)-(−)-N-acetylcolchinol via Ullmann biaryl coupling

Simon D. Broady, Michael Golden, John Leonard et al. · Tetrahedron Letters · 2007 · 42 citations

Cross-coupling Reaction, Asymmetric Synthesis, Organic Chemistry +2

Synthesis and structure-activity relationship of 4-(1,3-benzothiazol-2-yl)-thiophene-2-sulfonamides as cyclin-dependent kinase 5 (cdk5)/p25 inhibitors

Jonas Malmström, Jenny Viklund, Can Slivo et al. · Bioorganic & Medicinal Chemistry Letters · 2012 · 41 citations · Full text

Medicinal Chemistry, Heterocyclic, Medicine +13

New hydroxylamines for the synthesis of hydroxamic acids

Bernard Barlaam, A. Hamon, Mickaël Maudet · Tetrahedron Letters · 1998 · 33 citations

Engineering, New Hydroxylamines, Organic Chemistry +4