J. Martin Herold

Discovery of a 2,4-Diamino-7-aminoalkoxyquinazoline as a Potent and Selective Inhibitor of Histone Lysine Methyltransferase G9a

Feng Liu, Xin Chen, Abdellah Allali‐Hassani et al. · Journal of Medicinal Chemistry · 2009 · 236 citations · Full text

Molecular Biology, Chemical Biology, Pharmaceutical Chemistry +17

Protein Lysine Methyltransferase G9a Inhibitors: Design, Synthesis, and Structure Activity Relationships of 2,4-Diamino-7-aminoalkoxy-quinazolines.

Feng Liu, Xin Chen, Abdellah Allali‐Hassani et al. · Journal of Medicinal Chemistry · 2010 · 204 citations · Full text

Discovery of a chemical probe for the L3MBTL3 methyllysine reader domain

Lindsey I. James, Dalia Baršytė-Lovejoy, Nan Zhong et al. · Nature Chemical Biology · 2013 · 169 citations · Full text

Chemical Biology, Molecular Characterization, Natural Sciences +7

Optimization of Cellular Activity of G9a Inhibitors 7-Aminoalkoxy-quinazolines

Feng Liu, Dalia Baršytė-Lovejoy, Abdellah Allali‐Hassani et al. · Journal of Medicinal Chemistry · 2011 · 155 citations · Full text

Vitro Potency, Excellent Potency, Drug Target +16

Small-Molecule Ligands of Methyl-Lysine Binding Proteins

J. Martin Herold, Tim J. Wigle, Jacqueline L. Norris et al. · Journal of Medicinal Chemistry · 2011 · 119 citations · Full text