Tomoaki Koshizawa

Synthesis of 2,6-dimethyl-9-aryl-9-phosphabicyclo[3.3.1]nonanes: their application to asymmetric synthesis of chiral tetrahydroquinolines and relatives

Osamu Hara, Tomoaki Koshizawa, Kazuishi Makino et al. · Tetrahedron · 2007 · 38 citations

Engineering, Asymmetric Synthesis, Organic Chemistry +7

Synthesis of novel chiral 1,3-aminophenols and application for the enantioselective addition of diethylzinc to aldehydes

Xiaofeng Yang, Zhaohui Wang, Tomoaki Koshizawa et al. · Tetrahedron Asymmetry · 2007 · 22 citations

Engineering, Novel Chiral 1,3-Aminophenols, Organic Chemistry +7

Optimization of a novel series of potent and orally bioavailable GPR119 agonists

Tomoaki Koshizawa, Toshiharu Morimoto, Gen Watanabe et al. · Bioorganic & Medicinal Chemistry Letters · 2017 · 16 citations · Full text

Bioavailable Gpr119 Agonists, Pharmaceutical Science, Novel Series +8

Discovery of novel spiro[chromane-2,4′-piperidine] derivatives as potent and orally bioavailable G-protein-coupled receptor 119 agonists

Tomoaki Koshizawa, Toshiharu Morimoto, Gen Watanabe et al. · Bioorganic & Medicinal Chemistry Letters · 2018 · 12 citations · Full text

Medicinal Chemistry, Derivatives, Biochemistry +10

Discovery of a 2-hydroxyacetophenone derivative as an outstanding linker to enhance potency and β-selectivity of liver X receptor agonist

Minoru Koura, Yuki Yamaguchi, Sayaka Kurobuchi et al. · Bioorganic & Medicinal Chemistry · 2016 · 11 citations · Full text

2-Hydroxyacetophenone Derivative, Medicinal Chemistry, Pharmacological Study +10