Daniela Tomaselli

Novel polyamine-based Histone deacetylases-Lysine demethylase 1 dual binding inhibitors

Andrea Milelli, Chiara Marchetti, Eleonora Turrini et al. · Bioorganic & Medicinal Chemistry Letters · 2018 · 29 citations · Full text

Life Sciences, Molecular Biology, Pharmacology +12

Structure–Reactivity Relationships on Substrates and Inhibitors of the Lysine Deacylase Sirtuin 2 from <i>Schistosoma mansoni</i> ( <i>Sm</i> Sirt2)

Daria Monaldi, Dante Rotili, Julien Lancelot et al. · Journal of Medicinal Chemistry · 2019 · 25 citations · Full text

Life Sciences, Biochemistry, Medicinal Chemistry +17

Effect of α-Methoxy Substitution on the Anti-HIV Activity of Dihydropyrimidin-4(3<i>H</i>)-ones

Maxim B. Nawrozkij, Mariantonietta Forgione, A. S. Yablokov et al. · Journal of Medicinal Chemistry · 2018 · 22 citations

Pharmacy, Medicinal Chemistry, Pharmacology +11

Disruptor of telomeric silencing 1-like (DOT1L): disclosing a new class of non-nucleoside inhibitors by means of ligand-based and structure-based approaches

Manuela Sabatino, Dante Rotili, Alexandros Patsilinakos et al. · Journal of Computer-Aided Molecular Design · 2018 · 21 citations

Pharmacy, Medicinal Chemistry, Pharmacology +10

α,γ-Diketocarboxylic Acids and Their Esters Act as Carbonic Anhydrase IX and XII Selective Inhibitors

Alessio Nocentini, Alessia Lucidi, Francesca Perut et al. · ACS Medicinal Chemistry Letters · 2019 · 20 citations · Full text

Pharmacy, Medicinal Chemistry, Pharmacology +10