Concepedia
Statistics
Publications
17
Citations
765
H-Index
16
Active since
2014
Affiliations
University of California, Riverside(Current)
University of Milan
Sanford Burnham Prebys Medical Discovery Institute
University of California San Diego
Cedars-Sinai Medical Center
Luca Gambini is an author at University of California, Riverside specializing in medicine, pharmacology, and drug discovery.
Top concepts
MedicinePharmacologyDrug DiscoveryBiochemistryTumor BiologyNatural SciencesCancer BiologyChemical BiologyMedicinal ChemistryCell Biology
Publications per year
2014–2022
Covalent Inhibitors of Protein–Protein Interactions Targeting Lysine, Tyrosine, or Histidine Residues
Luca Gambini, Carlo Baggio, Parima Udompholkul et al. · Journal of Medicinal Chemistry · 2019 · 136 citations · Full text
Human resistin protects against endotoxic shock by blocking LPS–TLR4 interaction
Jessica Jang, Jiang Li, Luca Gambini et al. · Proceedings of the National Academy of Sciences · 2017 · 95 citations · Full text
Reduction of Circulating Cancer Cells and Metastases in Breast-Cancer Models by a Potent EphA2-Agonistic Peptide–Drug Conjugate
Ahmed F. Salem, Si Wang, Sandrine Billet et al. · Journal of Medicinal Chemistry · 2018 · 65 citations · Full text
NMR Fingerprints of the Drug‐like Natural‐Product Space Identify Iotrochotazine A: A Chemical Probe to Study Parkinson’s Disease
Tanja Grkovic, Rebecca H. Pouwer, Marie‐Laure Vial et al. · Angewandte Chemie International Edition · 2014 · 63 citations · Full text
Aryl-fluorosulfate-based Lysine Covalent Pan-Inhibitors of Apoptosis Protein (IAP) Antagonists with Cellular Efficacy
Carlo Baggio, Parima Udompholkul, Luca Gambini et al. · Journal of Medicinal Chemistry · 2019 · 60 citations · Full text
Protein Assembly, Apoptosis Protein, Apoptosis +19
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