Bastian Frehland

Synthesis and pharmacological evaluation of like- and unlike-configured tetrahydro-2-benzazepines with the α-substituted benzyl moiety in the 5-position

Peer Hasebein, Bastian Frehland, Kirstin Lehmkuhl et al. · Organic & Biomolecular Chemistry · 2014 · 75 citations

Pharmacy, Medicinal Chemistry, Pharmacology +13

Development of a selective competitive receptor binding assay for the determination of the affinity to NR2B containing NMDA receptors

Dirk Schepmann, Bastian Frehland, Kirstin Lehmkuhl et al. · Journal of Pharmaceutical and Biomedical Analysis · 2010 · 63 citations

Medicine, Medicinal Chemistry, Pharmacology +12

Conformationally constrained NR2B selective NMDA receptor antagonists derived from ifenprodil: Synthesis and biological evaluation of tetrahydro-3-benzazepine-1,7-diols

Bastian Tewes, Bastian Frehland, Dirk Schepmann et al. · Bioorganic & Medicinal Chemistry · 2010 · 62 citations · Full text

Pharmacy, Medicinal Chemistry, Pharmacology +14

Design, Synthesis, and Biological Evaluation of 3‐Benzazepin‐1‐ols as NR2B‐Selective NMDA Receptor Antagonists

Bastian Tewes, Bastian Frehland, Dirk Schepmann et al. · ChemMedChem · 2010 · 50 citations

Medicine, Medicinal Chemistry, Pharmacology +15

Enantiomerically Pure 2-Methyltetrahydro-3-benzazepin-1-ols Selectively Blocking GluN2B Subunit Containing <i>N</i>-Methyl-<scp>d</scp>-aspartate Receptors

Bastian Tewes, Bastian Frehland, Dirk Schepmann et al. · Journal of Medicinal Chemistry · 2015 · 39 citations

Medicine, Medicinal Chemistry, Pharmacology +10