Bertan Bopp

Targeting HSP90 dimerization via the C terminus is effective in imatinib-resistant CML and lacks the heat shock response

Sanil Bhatia, Daniela Diedrich, Benedikt Frieg et al. · Blood · 2018 · 79 citations · Full text

Medicine, Molecular Biology, Oncology +6

Naphthol AS-E Phosphate Inhibits the Activity of the Transcription Factor Myb by Blocking the Interaction with the KIX Domain of the Coactivator p300

Sagar Uttarkar, Sandeep Dukare, Bertan Bopp et al. · Molecular Cancer Therapeutics · 2015 · 70 citations · Full text

Life Sciences, Biochemistry, Molecular Biology +9

Development of a First-in-Class Small-Molecule Inhibitor of the C-Terminal Hsp90 Dimerization

Sanil Bhatia, Lukas V. Spanier, David Bickel et al. · ACS Central Science · 2022 · 35 citations · Full text

Medicine, Oncology, Pharmacology +14

Design and biological testing of peptidic dimerization inhibitors of human Hsp90 that target the C-terminal domain

Bertan Bopp, Emanuele Ciglia, Anissa Ouald-Chaib et al. · Biochimica et Biophysica Acta (BBA) - General Subjects · 2016 · 26 citations

Pharmacy, Medicinal Chemistry, Molecular Biology +14

Cryptotanshinone from Salvia miltiorrhiza Roots Reduces Cytokeratin CK1/10 Expression in Keratinocytes by Activation of Peptidyl-prolyl-cis-trans-isomerase FKBP1A

Stefan Esch, Simone König, Bertan Bopp et al. · Planta Medica · 2018 · 10 citations

Life Sciences, Biochemistry, Pharmacology +13