Elena Cendón

Hit to lead evaluation of 1,2,3-triazolo[4,5-b]pyridines as PIM kinase inhibitors

Joaquı́n Pastor, Julen Oyarzábal, Gustavo Saluste et al. · Bioorganic & Medicinal Chemistry Letters · 2012 · 44 citations · Full text

Pharmacy, Medicinal Chemistry, Pharmacology +12

Identification of ETP-46321, a potent and orally bioavailable PI3K α, δ inhibitor

Sonia Martı́nez, Ana Isabel Hernández, Carmen Varela et al. · Bioorganic & Medicinal Chemistry Letters · 2012 · 24 citations · Full text

Pharmacy, Medicinal Chemistry, Pharmacology +11

Rapid identification of ETP-46992, orally bioavailable PI3K inhibitor, selective versus mTOR

Sonia Martı́nez, Ana Isabel Hernández, Carmen Varela et al. · Bioorganic & Medicinal Chemistry Letters · 2012 · 19 citations · Full text

Pharmacy, Medicinal Chemistry, Pharmacology +12

Generation of tricyclic imidazo[1,2-a]pyrazines as novel PI3K inhibitors by application of a conformational restriction strategy

Sonia Martı́nez, Sonsoles Rodríguez-Arístegui, Ana Isabel Hernández et al. · Bioorganic & Medicinal Chemistry Letters · 2017 · 10 citations · Full text

Pharmacy, Medicinal Chemistry, Pharmacology +14