Modulation of the Heparanase-inhibiting Activity of Heparin through Selective Desulfation, Graded N-Acetylation, and Glycol Splitting

Annamaria Naggi, Benito Casu, Marta Pérez, +7

Journal of Biological Chemistry

The 4-hydroxybenzoate/4-aminophenazone chromogenic system used in the enzymic determination of serum cholesterol.

F Meiattini, L Prencipe, Fabrizio Bardelli, +2

Clinical Chemistry

Lipid AnalysisCholesterol EsteraseEnzymic DeterminationSerum CholesterolBioanalysis +14

Heterocyclic and Phenyl Double-Bond-Locked Combretastatin Analogues Possessing Potent Apoptosis-Inducing Activity in HL60 and in MDR Cell Lines

Daniele Simoni, Giuseppina Grisolia, Giuseppe Giannini, +17

Journal of Medicinal Chemistry

Novel Combretastatin Analogues Endowed with Antitumor Activity

Daniele Simoni, Romeo Romagnoli, Riccardo Baruchello, +12

Journal of Medicinal Chemistry

Undersulfated and Glycol-Split Heparins Endowed with Antiangiogenic Activity

Benito Casu, Marco Guerrini, Sara Guglieri, +12

Journal of Medicinal Chemistry

GlycobiologyImmunologyEpoxide RingsTumor BiologyAngiogenesis +18

Biological and molecular properties of a new αvβ3/αvβ5 integrin antagonist

Laura Belvisi, Teresa Riccioni, Marcella Marcellini, +16

Molecular Cancer Therapeutics

Synthesis and Evaluation of New Hsp90 Inhibitors Based on a 1,4,5-Trisubstituted 1,2,3-Triazole Scaffold

Maurizio Taddei, Serena Ferrini, Luca Giannotti, +15

Journal of Medicinal Chemistry

Molecular DockingMedicinal ChemistryBiochemistryCompound 18Drug Discovery +12

Potent Integrin Antagonists from a Small Library of RGD-Including Cyclic Pseudopeptides

Laura Belvisi, Anna Bernardi, Anna Checchia, +7

Organic Letters

Peptide EngineeringRgd-including Cyclic PseudopeptidesPharmacotherapyChemical BiologyPharmaceutical Chemistry +15

Short Heparin Sequences Spaced by Glycol-Split Uronate Residues Are Antagonists of Fibroblast Growth Factor 2 and Angiogenesis Inhibitors

Benito Casu, Marco Guerrini, Annamaria Naggi, +10

Biochemistry

Fgf2 DimerizationAngiogenesis InhibitorsGlycobiologyFibroblast Growth Factor-2Angiogenesis +19

Synthesis and Biological Activity of Fluorinated Combretastatin Analogues

Domenico Alloatti, Giuseppe Giannini, Walter Cabri, +10

Journal of Medicinal Chemistry

Combinatorial ChemistryMedicinal ChemistryBioorganic ChemistryFluorinated Combretastatin AnaloguesBiochemistry +13