Concepedia
Statistics
Publications
6
Citations
134
H-Index
Active since
2014
Affiliations
La Trobe University(Current)
Monash University
Burnet Institute
The University of Melbourne
New York University
Melissa J. Buskes is an author at La Trobe University specializing in medicinal chemistry, drug discovery, and medicine.
Top concepts
MedicinePharmacologyDrug DiscoveryMedicinal ChemistryMalariaBiochemistryChemical BiologyDrug DevelopmentNatural Sciences
Publications per year
2014–2020
Improvement of Aqueous Solubility of Lapatinib-Derived Analogues: Identification of a Quinolinimine Lead for Human African Trypanosomiasis Drug Development
Kelly A. Bachovchin, Amrita Sharma, Seema Bag et al. · Journal of Medicinal Chemistry · 2018 · 36 citations · Full text
A 4-cyano-3-methylisoquinoline inhibitor of Plasmodium falciparum growth targets the sodium efflux pump PfATP4
Paul R. Gilson, Rasika Kumarasingha, Jennifer K. Thompson et al. · Scientific Reports · 2019 · 31 citations · Full text
Scaffold and Parasite Hopping: Discovery of New Protozoal Proliferation Inhibitors
Baljinder Singh, Jean Bernatchez, Laura‐Isobel McCall et al. · ACS Medicinal Chemistry Letters · 2020 · 26 citations · Full text
Antimalarial activity of novel 4-cyano-3-methylisoquinoline inhibitors against Plasmodium falciparum: design, synthesis and biological evaluation
Melissa J. Buskes, Katherine Harvey, Benjamin J. Richards et al. · Organic & Biomolecular Chemistry · 2016 · 17 citations
Synthesis and biological evaluation of 2-anilino-4-substituted-7H-pyrrolopyrimidines as PDK1 inhibitors
Nathan J. O’Brien, Martin Brzozowski, Melissa J. Buskes et al. · Bioorganic & Medicinal Chemistry · 2014 · 12 citations · Full text
Medicinal Chemistry, Medicine, Pdk1 Inhibitors +3
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