Stephen L. Garland

Definition of the G Protein-Coupled Receptor Transmembrane Bundle Binding Pocket and Calculation of Receptor Similarities for Drug Design

David E. Gloriam, Steven M. Foord, Frank E. Blaney et al. · Journal of Medicinal Chemistry · 2009 · 97 citations

Medicine, Molecular Biology, Pharmacology +17

(1H-Imidazo[4,5-c]pyridin-2-yl)-1,2,5-oxadiazol-3-ylamine derivatives: A novel class of potent MSK-1-inhibitors

Mark J. Bamford, Michael J. Alberti, Nicholas Bailey et al. · Bioorganic & Medicinal Chemistry Letters · 2005 · 43 citations · Full text

Pharmacy, Medicinal Chemistry, Pharmacology +5

Non-peptidic antagonists of the CGRP receptor, BIBN4096BS and MK-0974, interact with the calcitonin receptor-like receptor via methionine-42 and RAMP1 via tryptophan-74

Philip S. Miller, James Barwell, David R. Poyner et al. · Biochemical and Biophysical Research Communications · 2009 · 41 citations · Full text

Medicine, Pharmacology, Pharmacotherapy +17

Design criteria for molecular mimics of fragments of the β-turn. 1. Cα atom analysis

Stephen L. Garland, P. M. Dean · Journal of Computer-Aided Molecular Design · 1999 · 29 citations

Pharmacy, Chemistry, Medicinal Chemistry +16

The identification of structurally novel, selective, orally bioavailable positive modulators of mGluR2

Pier Luca D’Alessandro, Corrado Corti, Adelheid Roth et al. · Bioorganic & Medicinal Chemistry Letters · 2009 · 23 citations · Full text

Pharmacy, Medicinal Chemistry, Pharmacology +8