Design, synthesis, modeling studies and biological screening of novel pyrazole derivatives as potential analgesic and anti-inflammatory agents

Azza T. Taher, Marwa T. Sarg, Nermeen R. El-Sayed Ali, +1

Bioorganic Chemistry

Medicinal ChemistryAnti-inflammatory AgentsBiochemistryNovel Pyrazole DerivativesMedicine +8

Pimenta dioica (L.) Merr. Bioactive Constituents Exert Anti-SARS-CoV-2 and Anti-Inflammatory Activities: Molecular Docking and Dynamics, In Vitro, and In Vivo Studies

Heba A. El Gizawy, Sylvia A. Boshra, Ahmed Mostafa, +5

Molecules

Novel 1,3,4-heterodiazole analogues: Synthesis and in-vitro antitumor activity

Azza T. Taher, Hanan H. Georgey, Hussein I. El‐Subbagh

European Journal of Medicinal Chemistry

Medicinal ChemistryMedicineNovel 1,3,4-Heterodiazole AnaloguesAnti-cancer AgentHeterocycle Chemistry +3

Newly synthesized series of oxoindole–oxadiazole conjugates as potential anti-SARS-CoV-2 agents:<i>in silico</i>and<i>in vitro</i>studies

Rana M. El-Masry, Ahmed A. Al‐Karmalawy, Radwan Alnajjar, +5

New Journal of Chemistry

Molecular Pharmacology1,3,4-Oxadiazole–oxoindole ConjugatesAntiviral CompoundMedicineAntiviral Drug Development +10

Synthesis of novel isatin-thiazoline and isatin-benzimidazole conjugates as anti-breast cancer agents

Azza T. Taher, Nadia A. Khalil, Eman Ahmed

Archives of Pharmacal Research

MedicineIsatin-benzimidazole ConjugatesPharmacotherapyAnti-cancer AgentDrug Development +4

Design, synthesis and cytotoxic activity of certain novel chalcone analogous compounds

Salwa Elmeligie, Azza T. Taher, Aliaa M. Kamal, +1

European Journal of Medicinal Chemistry

MedicineChemistryHeterocycle ChemistryCytotoxic ActivityPharmacology +3

Synthesis and Bioactivity Evaluation of New 6-Aryl-5-cyano Thiouracils as Potential Antimicrobial and Anticancer Agents

Azza T. Taher, Sahar M. Abou‐Seri

Molecules

B. SubtilisNew 6-Aryl-5-cyano ThiouracilsAnticancer AgentsAntimicrobial ChemotherapyChemistry +20

Alkoxyphenylthiazoles with broad-spectrum activity against multidrug-resistant gram-positive bacterial pathogens

Moustafa ElAwamy, Haroon Mohammad, Abdelrahman Hussien, +7

European Journal of Medicinal Chemistry

Health SciencesAntibioticsMedicineBroad-spectrum ActivityAntibacterial Agent +7

Synthesis and in-vitro anti-proliferative evaluation of some pyrazolo[1,5-a]pyrimidines as novel larotrectinib analogs

Mohamed H. Attia, Eman Z. Elrazaz, Soad Z. El‐Emam, +3

Bioorganic Chemistry

In-vitro Anti-proliferative EvaluationMedicinal ChemistryPharmaceutical ScienceBioorganic ChemistryBiochemistry +9

Evaluation of N-phenyl-2-aminothiazoles for treatment of multi-drug resistant and intracellular Staphylococcus aureus infections

Inas G. Shahin, Nader S. Abutaleb, Marwa Alhashimi, +5

European Journal of Medicinal Chemistry

Multi-drug ResistantAntibiotic AdjuvantPharmacologyPharmacotherapyAntibacterial Agent +6